Synthesis of Tetrazolo, Triazolo and Quinazolino Annulated Analogues of the Privileged Nucleus of Pyrrolo-[1, 5]-Benzothiazepines of Medicinal Interest
Journal Title: International Journal of Scientific Research and Reviews - Year 2013, Vol 2, Issue 2
Abstract
The nucleophilic displacement of 2-iminothiomethylether derivative of pyrrolo-1,5- benzothiazepines was elegantly exploited in its reaction with bidentate nucleophiles such as NH2-NH2 (followed by reaction with HNO2), acetahydrazide, isatoic anhydride, amino benzonitrile to allow the facile annulation of this molecule with triazole, tetrazole and quinazoline nucleus.
Authors and Affiliations
Priyanka Rani , D. Kishore
Keywords
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