SYNTHESIS AND ANTIMICROBIAL EVALUATION OF SOME AMINO ACID DERIVATIVES OF 2-AMINO-4-METHYLTHIAZOLE
Journal Title: Analele Universitatii din Bucuresti. Chimie - Year 2010, Vol 19, Issue 2
Abstract
The synthesis of a new series of 2-[N-(Tos-, Pht- or tetrachlorophthalyl)-aminoacyl]- or free 2-(aminoacyl)- or 2-[N-(Tos- or Pht-)dipeptidyl]amino-4-methyl-thiazole derivatives (II-XXIII) is described. Further, Schiff base and hippuroyl compounds (XXIV and XXV respectively) are obtained in high yield. The biological activity of the compounds cited in this article is reported.
Authors and Affiliations
H. M. Hassan, A. F. El-Haddad, F. A. Kora, A. M. El-Naggar
Keywords
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